- 英文名称
- [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
- 分子式
- C183H281N57O54S2
- 分子量
- 4207.67
- 中文别名
- 化合物[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide; (GLY1,SER3·22,GLN4·34,THR6,ARG19,TYR21,ALA23·31,AIB32)-人胰多肽; [CPP1-7,NPY19-23,ALA31,AIB32,GLN 34]-胰多肽; 神经肽YY5受体激动剂多肽; (Gly1,Ser3·22,Gln4·34,Thr6,Arg19,Tyr21,Ala23·31,Aib32)-Pancreatic Polypeptide (human); (Gly1,Gln4·16,Thr6·13,Tyr7,Asp10,Asn11,Pro14,Arg26,Met30,Ala31,Aib32)-Neuropeptide Y (human, rat); H-Gly-Pro-Ser-Gln-Pro-Thr-Tyr-Pro-Gly-Asp-Asn-Ala-Thr-Pro-Glu-Gln-Met-Ala-Arg-Tyr-Tyr-Ser-Ala-Leu-Arg-Arg-Tyr-Ile-Asn-Met-Ala-Aib-Arg-Gln-Arg-Tyr-NH2; Glycyl-L-prolyl-L-seryl-L-glutaminyl-L-prolyl-L-threonyl-L-tyrosyl-L-prolylglycyl-L-α-aspartyl-L-asparaginyl-L-alanyl-L-threonyl-L-prolyl-L-α-glutamyl-L-glutaminyl-L-methionyl-L-alanyl-L-arginyl-L-tyrosyl-L-tyrosyl-L-seryl-L-alanyl-L-leucyl-L-arginyl-L-arginyl-L-tyrosyl-L-isoleucyl-L-asparaginyl-L-methionyl-L-alanyl-2-methylalanyl-L-arginyl-L-glutaminyl-L-arginyl-L-tyrosinamide
- 用途
- 有效的选择性神经肽YY5受体激动剂,与hY5受体结合的IC50值为0.24nM;增加饮食摄入量;在成年雄性大鼠中以剂量依赖性方式诱导大量食物摄入