10605-03-5 2,3,9,10-四甲氧基-13-甲基-5,6-二氢异喹啉并[3,2-α]异喹啉-7-氯化物
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安全说明
运输方式为冰袋运输。危险性质:非危险化学品。海关编码:2933399990。毒性数据:小鼠静脉注射LD50为9500ug/kg(9.5mg/kg),来源为美国专利文献第3849561号。
用途与制备
Dehydrocorydaline chloride (13-Methylpalmatine chloride) is a bioactive alkaloid from Corydalis yanhusuo. It regulates Bax/Bcl-2 expression, activates caspases-7/-8, inactivates PARP, enhances p38 MAPK activation, and has anti-inflammatory, anti-cancer, and potent antimalarial effects (IC50=38 nM for P. falciparum 3D7). In vitro, it promotes muscle differentiation and inhibits MCF-7 proliferation via apoptosis. In vivo, it shows dose-dependent antinociceptive effects in mice.
生命科学; 中草药成分; 医药