作为医药中间体，用于相关药物的合成制备。
医药
合成路线 1（1. 合成：76360-82-2）
产率：100%
合成条件：at 0℃; for 0.50 h;
实验步骤：在0℃下，将EtOH中的甲胺（33％，17.5mL，140mmol）缓慢加入到中间体3（10.0g，43.1mmol）在120mL二氯甲烷中的溶液中。 将溶液搅拌30分钟。 加入水（150ml），分离所得混合物，用MgSO 4干燥有机层，过滤，浓缩，得到标题化合物（9.77g，100％），为白色固体。
参考文献：
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