作为医药中间体，用于相关药物分子的合成（具体用途需结合具体药物研发背景）。
医药
合成路线 1（1. 合成：53631-18-8）
产率：83%
合成条件：With Oxone; ammonium bromide In methanol for 2 h; Reflux
实验步骤：通用方法：将Oxone（1.352g，2.2mmol）加入到充分搅拌的底物（2mmol）和NH 4 Br（0.215g，2.2mmol）的甲醇（10ml）溶液中，并将反应混合物在室温下搅拌 （或回流温度）。 通过TLC监测反应完成后，将反应混合物用硫代硫酸钠水溶液淬灭，并用乙酸乙酯（3.x.25ml）萃取。 最后，将合并的有机层用水洗涤，用无水硫酸钠干燥，过滤并真空除去溶剂，得到粗残余物，将其通过硅胶柱色谱（细于200目）进一步纯化，得到纯产物。 所有产物均在1H NMR和质谱数据的基础上鉴定。
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