作为有机合成中间体，广泛应用于医药领域的相关化合物合成。
医药
合成路线 1（1. 合成：144072-29-7）
- 步骤: 向对氨基-苯甲醇（1g，8.12mmol，1当量）在80mL无水THF中的溶液中加入DIEA（1.4mL，8.12mmol，1当量）和Boc₂O（1.9mL，8.12mmol，1当量）；将混合物加热至回流过夜，冷却并真空蒸发；残余物溶于EtOAc，用0.1N HCl洗涤，MgSO₄干燥，过滤并真空蒸发；硅胶柱色谱（Hex-EtOAc，1:1）纯化得产物。
- 条件: With N-ethyl-N,N-diisopropylamine In tetrahydrofuran; Heating / reflux
- 产率: 100%
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